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10 resultsUpdated October 25, 2026
1

Estradiol contributes to sex differences in resilience to sepsis-induced metabolic dysregulation and dysfunction in the heart via GPER-1-mediated PPARδ/NLRP3 signaling

Metabolism 156 (2024)

Joseph Adu-Amankwaah; Adebayo Oluwafemi Adekunle; Ziqing Tang; Aisha Bushi; Rubin Tan; Lu Fu; Zheng Gong; Ziyu Ma; Richard Mprah; Marie Louise Ndzie Noah; Prosperl Ivette Wowui; Jeremiah Ong'achwa Machuki; Xiuhua Pan; Tao Li; Hong Sun

2

G protein-coupled estrogen receptor biased signaling in health and disease

Pharmacology & Therapeutics 269 (2025)

Aisha Bushi; Yixuan Ma; Joseph Adu-Amankwaah; Rong Wang; Fen Cui; Rui Xiao; Jinming Zhao; Jinxiang Yuan; Rubin Tan

3

Cardioprotective effects of GPER agonist in ovariectomized diabetic rats: reversing ER stress and structural changes

Naunyn-Schmiedeberg's Archives of Pharmacology 398(3) (2025)

Mohammad Amin Ghaffari Sirizi; Mansour Esmailidehaj; Seyed-Mahdi Mohamadi-Zarch; Maryam Yadeghari; Hossein Azizian

4

Pharmacological Stimulation of GPER Reverses Mitochondrial Dysfunction in the Hearts of Ovariectomized Type 2 Diabetic Rats

Journal of Biochemical and Molecular Toxicology 39(12) (2025)

Nahlah Fahad‐Alreshidi; Refaat A. Eid; Abdullah M. K. Albloshi; Saud S. Alharbi; Sultan Mohammed Alanazi; Thamer Alsufayan; Musaad B. Alsahly; Mirwais Ramozi

5

The G protein-coupled oestrogen receptor GPER in health and disease: an update

Nature Reviews Endocrinology 19(7) (2023)

Eric R. Prossnitz; Matthias Barton

6

GPER in metabolic homeostasis and disease: molecular mechanisms, nutritional regulation, and therapeutic potential

Journal of Translational Medicine 23(1) (2025)

Liyan Liu; Yutao Zhou; Jing Liu; Xinmiao Zhang; Chongwu He; Xiaoqiang Zeng; Rebeka Dejenie; Usman Zeb; Qiao Zeng; Lan Liu; Jianglong Li; Xingsheng Zeng; Qinglong Hu; Xianming Huang; Xue Xu; Hanzhi Dong; Jinxiu Zhong; Yanxiao Huang; Qiaoli Lv; Bo Liu; Yu-an Qiu; Tenghua Yu

7

GPER activation attenuates cardiac dysfunction by upregulating the SIRT1/3-AMPK-UCP2 pathway in postmenopausal diabetic rats

PLOS ONE 18(12) (2023)

Hossein Azizian; Zeinab Farhadi; Michael Bader; Jalil Alizadeh Ghalenoei; Mohammad Amin Ghafari; Shokoufeh Mahmoodzadeh; Meijing Wang

8

Puerarin 6″-O-xyloside improves postmenopausal lipid metabolic disorders via the PPARα-mediated FAO pathway

Phytomedicine 152 (2026)

Danna Wang; Yalin You; Tianyu Luo; Tingting Chen; Xiaoqin Wu; Jiawen Huang; Yong Gao; Guangning Nie

9

Selective ERα Attenuates Hypothalamic ER Stress and Regulates Energy Homeostasis in Ovariectomized Mice Fed With High‐Fat Diet

Journal of Biochemical and Molecular Toxicology 39(9) (2025)

Amr Ali Mohamed Abdelgawwad El‐Sehrawy; Amirhosseinjaberi; Ehsan Zandi; Farzaneh Yazdi; Setarehsadat Rafiei; Ibrokhim Sapaev; Sepideh KarkonShayan; Payam Ali Khiavi; Pouria Salajegheh; Melina Shadi; Reza Akhavan‐Sigari

10

Estrogen, Epigenetics, and Cardiometabolic Health: Mechanisms and Therapeutic Strategies in Postmenopausal Women

Cells 15(6) (2026)

Ailene Edwards; Pranjal Singh; Vyan Shah; Vivek Chander; Sumita Mishra