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81 resultsUpdated October 25, 2026
1

Different applications of machine learning approaches in materials science and engineering: Comprehensive review

Engineering Applications of Artificial Intelligence 135 (2024)

Yan Cao; Ali Taghvaie Nakhjiri; Mahdi Ghadiri

2

The Effect of the Particle Size Reduction on the Biorelevant Solubility and Dissolution of Poorly Soluble Drugs with Different Acid-Base Character

Pharmaceutics 15(1) (2023)

Dóra Csicsák; Rita Szolláth; Szabina Kádár; Rita Ambrus; Csilla Bartos; Emese Balogh; István Antal; István Köteles; Petra Tőzsér; Vivien Bárdos; Péter Horváth; Enikő Borbás; Krisztina Takács‐Novák; Bálint Sinkó; Gergely Völgyi

3

Recent developments in the use of nanocrystals to improve bioavailability of APIs

Wiley Interdisciplinary Reviews Nanomedicine and Nanobiotechnology 16(2) (2024)

Yidan Ding; Tongyi Zhao; Jianing Fang; Jiexin Song; Haobo Dong; Jiarui Liu; Sijin Li; Min Zhao

4

Sugars and Polyols of Natural Origin as Carriers for Solubility and Dissolution Enhancement

Pharmaceutics 15(11) (2023)

Madan Poka; Marnus Milne; Anita Wessels; Marique Elizabeth Aucamp

5

Emerging role of nanocrystals in pharmaceutical applications: A review of regulatory aspects and drug development process

Applied Materials Today 40 (2024)

Padakanti Sandeep Chary; Samia Shaikh; Valamla Bhavana; Naveen Rajana; Ravindra Vasave; Neelesh Kumar Mehra

7

Towards the prediction of drug solubility in binary solvent mixtures at various temperatures using machine learning

Journal of Cheminformatics 16(1) (2024)

Zeqing Bao; Gary Tom; Austin Cheng; Jeffrey Watchorn; Alán Aspuru‐Guzik; Christine J. Allen

9

Choline-Amino Acid-Derived Bio-ionic Liquids for Solubility Enhancement of Zafirlukast

AAPS PharmSciTech 23(5) (2022)

Namrata Gaikwad; Swapna Kudal; Amelia M. Avachat

10

Third-Generation Solid Dispersion Through Lyophilization Enhanced Oral Bioavailability of Resveratrol

ACS Pharmacology & Translational Science 7(3) (2024)

Hugo Almeida; Bárbara Ferreira; Carlos Fernandes‐Lopes; Francisca Araújo; Maria João Bonifácio; Teófilo Vasconcelos; Bruno Filipe Carmelino Cardoso Sarmento

11

Biofunctional Excipients: Their Emerging Role in Overcoming the Inherent Poor Biopharmaceutical Characteristics of Drugs

Pharmaceutics 17(5) (2025)

Milad Reda Qelliny; Wesam W. Mustafa; Adel M. Al Fatease; Ali H. Alamri; Raid Ghassan Alany; Hamdy Abdelkader

12

Solubility enhancement of caffeine and furosemide using deep eutectic solvents formed by choline chloride and xylitol, citric acid, sorbitol or glucose

Journal of Drug Delivery Science and Technology 79 (2022)

Laura Lomba; Alejandra Polo; Julia Alejandre; Nuria Martínez; Beatriz Giner

13

Ibuprofen solubility and cytotoxic study of deep eutectic solvents formed by xylitol, choline chloride and water

Journal of Drug Delivery Science and Technology 82 (2023)

Laura Lomba; Ma Pilar Garralaga; Álvaro Werner; Beatriz Giner; Pedro M. Baptista; Natalia Sánchez‐Romero

14

Deep eutectic solvents based on sugars for oral applications

European Journal of Pharmaceutics and Biopharmaceutics 191 (2023)

Laura Lomba; Alejandra Polo; Álvaro Werner; Carlos Lafuente; Beatriz Giner

15

Nanocrystals: A Deep Insight into Formulation Aspects, Stabilization Strategies, and Biomedical Applications

Recent Patents on Nanotechnology 17(4) (2022)

Parijat Pandey; Deepika Purohit; S.K. Sharma; Avneet Kaur Lamba; Sapna Saini; Neha Minocha; Neelam Vashist; Dhirender Kaushik

16

A Comparison of Spray-Drying and Co-Precipitation for the Generation of Amorphous Solid Dispersions (ASDs) of Hydrochlorothiazide and Simvastatin

Journal of Pharmaceutical Sciences 112(8) (2023)

Monika Myślińska; Michael W. Stocker; Steven Ferguson; Anne Marie Healy

17

Solubility behavior of Rosiglitazone in ten pure solvents: Model correlation, thermodynamic calculations, and molecular simulation

Journal of Molecular Liquids 417 (2024)

Xiaojie Zhou; Aoran Xiong; Yuxi Zhen; Yizhen Yan; Xiangyang Zhang

18

Enhancing the dissolution and bacteriostatic activity of trimethoprim through salt formation

CrystEngComm 25(23) (2023)

Xingchen Hu; Yuntian Xiao; Luguang Qi; Yunhe Bai; Ying Ji Sun; Yang Ye; Chuang Xie

19

Physical stability and dissolution of ketoprofen nanosuspension formulation: Polyvinylpyrrolidone and Tween 80 as stabilizers

Pharmacia 70(1) (2023)

TENGKU ISMANELLY HANUM; Azizah Nasution; Sumaiyah Sumaiyah; Hakim Bangun

20

CFD modelling and simulations of atomization-based processes for production of drug particles: A review

International Journal of Pharmaceutics 670 (2025)

Mohamad Baassiri; Vivek Vinayak Ranade; Luís Padrela

21

Microwave-assisted, sulfhydryl-modified β-cyclodextrin-silymarin inclusion complex: A diverse approach to improve oral drug bioavailability via enhanced mucoadhesion and permeation

Carbohydrate Polymers 348(Pt B) (2024)

Shumaila Arshad; Syed Atif Raza; Alamgeer; Syed Nasir Abbas Bukhari; Nasser Fahad Alotaibi; Naveed Ahmad; Hafiz Muhammad Irfan; Arshad Mahmood; Mulazim Hussain Asim

22

Cocrystal Engineering-Based Strategies for Enhancing the Permeability of Poorly Permeable APIs

Crystal Growth & Design 25(18) (2025)

Maan Singh; Mayuri P. Sawarkar; Madhukiran R. Dhondale; Dolores R. Serrano; Ashish Kumar Agrawal; Dinesh K. Kumar

23

A comprehensive review of green approaches to drug solubility enhancement

Drug Development and Industrial Pharmacy 51(7) (2025)

B S Mahesha; F R Sheeba; H. K. Deepak

24

A Comprehensive Review of Solubility Enhancement Techniques for Poorly Soluble Drugs

Journal of Solution Chemistry 55(2) (2025)

Rajeswari Saripilli; Dinesh Kumar Sharma

25

Development and Characterization of Polymeric Films Loaded with Terbinafine for Fungal Infection Treatment

Polymers 17(8) (2025)

Gabriela Biliuță; Simona Gherman; Raluca Ioana Baron; Alexandra Bargan; Lăcrămioara Ochiuz; Cristina Tuchiluş; A Spac; Daniela Elena Zavastin

26

Therapeutic Potential of 2,2′:6′,2″-Terpyridine-Based Au(III), Pt(II), and Mn(II) Complexes against 2D and 3D Human Colorectal Resistant Cancer Cells

Journal of Medicinal Chemistry 68(21) (2025)

Katarzyna Choroba; B. Machura; Mateusz Penkala; Karol Erfurt; Sandra Zorat Cordeiro; Vanessa Araújo; Edvânia Leopoldo; Rute Lima; Diogo Afonso; Pedro Viana Baptista; Alexandra Ramos Fernandes

27

Cocrystals of antibiotics: enhancing antimicrobial efficacy through crystal engineering

Chemical Papers 79(5) (2025)

Amin Alvani; Ali Shayanfar; Raha Kaviani

29

Cationic surfactants: Fundamental aspects and functionality in the light of petrochemical industry challenges

Journal of Molecular Liquids 439 (2025)

Gulnara A. Gaynanova; Leysan A. Vasileva; Е. А. Романова; Lucia Ya. Zakharova; Oleg Gerol'dovich Sinyashin

30

A Scalable Freeze-Dissolving Approach to Prepare Ultrafine Crystals for Inhalation: Mechanism and Validation

Crystal Growth & Design 24(7) (2024)

Shengzheng Guo; Yuechao Cao; Yuxin Zhang; Yan Wang; Zhenguo Gao; Junbo Gong

31

Computational Modelling for Formulation Design

Springer eBooks (2025)

Teja Kumar Ponduri; Roja Rani Budha; Deepika Paliwal; Kartheek Siripurapu; Rajasekhar Reddy Alavala; GSN Koteswara Rao

34

Mathematical optimization and prediction of Febuxostat xanthine oxidase inhibitor solubility through supercritical CO2 system using machine-learning approach

Journal of Molecular Liquids 387 (2023)

Umme Hani; Zainab Ali Bu sinnah; Ahmad J. Obaidullah; Jowaher Alanazi; Muteb Alanazi; Tareq Nafea Alharby; Ahmed Abdullah Al Awadh; Ahmed A. Lahiq

35

Recent Developments In Brain-Targeted Drug Delivery Systems via Intranasal Route

Farmacja Polska 78(12) (2023)

Ahmad Ainurofiq; Aji Prasetya; Bingah Ginanjar Rahayu; Muhammad Syayiq Al Qadri; Myrat Kovusov; Ophira Evangelista Putri Laksono

36

Factors affecting the preparation of Cilnidipine nanoparticles

Iraqi Journal of Pharmaceutical Sciences 32(Suppl.) (2023)

Ruaa A. ALZALZALEE; Hanan Kassab

37

Design of Etched- and Functionalized-Halloysite/Meloxicam Hybrids: A Tool for Enhancing Drug Solubility and Dissolution Rate

Pharmaceutics 16(3) (2024)

Valeria Friuli; Claudia Urru; Chiara Ferrara; Debora Maria Conti; Giovanna Bruni; Lauretta Maggi; Doretta Capsoni

38

Chitosan as floating-mucoadhesive polymers in gastroretentive drug delivery

Science, Engineering and Health Studies (2023)

Ahmad Ainurofiq; Adinda Putri Febrina Sari; Ana Mardhiyah; Fauziyyah Sakinatun Nisa; Rahma Luthfiani Azka; Salsabilla Kania Putri; Vidiya Listiyani Saputri

39

New salts of teriflunomide (TFM) – Single crystal X-ray and solid state NMR investigation

Solid State Nuclear Magnetic Resonance 122 (2022)

Tomasz Pawlak; Piotr Paluch; Rafał Dolot; Grzegorz Bujacz; Marek J. Potrzebowski

40

Low-melting mixture solvents as novel solubilizing agents: Improving tolvaptan formulation and therapeutic efficacy

Journal of Molecular Liquids 414 (2024)

Xiuxiu Huang; Wenqing Dong; Xiao Luo; Lu Xu; Dongzhi Yang; Yinan Wang

42

Development and Characterization of an Ibuprofen-Salicylic Acid Co-crystal with Improved Solubility

Journal of Pharmaceutical Innovation 20(2) (2025)

Sonal Dubey; T Dheerathi; Dilip R. Reddy; Manisha Rajou

43

A Comprehensive Review on Polycaprolactone: A Promising Polymer for Enhancing Drug Bioavailability

Polymer-Plastics Technology and Materials 64(13) (2025)

Swati Dubey; Sanjeev Patel; Madhulika Pradhan; Krishna Yadav; Sunita Minz

44

Oligoethylene Phosphoramidate‐Based Kinase Inhibitor Prodrugs – Solubility, Enzyme Inhibition, and Hydrolysis

Chemistry - A European Journal 31(12) (2025)

Sarah Spiewok; Maximilian Schaefer; Markus Lamla; Yannick Jaritz; Alexander J. C. Kuehne

45

Experimental screening and molecular dynamics simulation study on wetting agent in dry suspension

Journal of Drug Delivery Science and Technology 95 (2024)

Minfang Feng; Yuting Tian; Yingying Zhang; Cuiting Yang; Xinhui Peng; Shuai Cen; Mengke Sheng; Zhixun Li; Qing Zhou; Xingxing Dai; Xinyuan Shi

46

Unveiling the role of solubilization of metformin hydrochloride assimilated in nonionic surfactants mediated mixed micellar assemblies

Colloids and Surfaces A Physicochemical and Engineering Aspects 703 (2024)

Nida Fatima; Muhammad Usman; Amnah Yusaf; Tanveer Hussain Bokhari; Nadia Akram; Saima Rehman; Sajjad Haider; Muhammad Siddiq; Muhammad Ahsan Bhatti; Mohammad Arif Cheema

47

A Quaternary Solid Dispersion System for Improving the Solubility of Olaparib

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Tae-Han Yun; Jeong-Gyun Lee; Kyu-Ho Bang; Jung Hyun Cho; Kyeong Soo Kim

48

Validation of UV spectrophotometric method for ketoprofen multicomponent crystals with malic acid and tartaric acid

Journal of Physics Conference Series 2190(1) (2022)

C F S Syamdini; I K Muthiah; Ahmad Ainurofiq

49

Solubility Enhancement, Formulation and Evaluation of Solid Tablet of Tinidazole

Indian Journal of Health Care Medical & Pharmacy Practice 4(2) (2023)

Ashutosh SHARMA; Ravi Kumar; Sunil Kumar; Yogesh Kumar Sharma; Surbhi Jangir

50

A Phosphoramidate Prodrug Platform: One‐Pot Amine Functionalization of Kinase Inhibitors with Oligoethylene Glycol for Improved Water‐Solubility

Chemistry - A European Journal 30(49) (2024)

Sarah Spiewok; Markus Lamla; Maximilian Schaefer; Alexander J. C. Kuehne

51

Review: Solid Dispersion Formulation Methods and Applications in Drug Delivery

Current Physical Chemistry 15(2) (2024)

Neelam Sihag; Kavita Bahmani; Samiksha Grewal; Rajni Tanwar; Nisham Rani; Jyoti Malik; Sunita Devi

53

Principal component analysis (PCA) of bioactive compounds and antioxidant activity of various sample particle sizes of sea urchin shells from coastal area of Lombok Island

Research Journal of Pharmacy and Technology (2024)

Legis Ocktaviana Saputri; Nurhidayati Nurhidayati; Herpan Syafii Harahap; Fitriannisa Faradina Zubaidi; Arina Windri Rivarti; Lina Permatasari

54

Various Aspects of Solid Dispersion Technology: A Review

Research Journal of Pharmacy and Technology (2025)

Deepika Sharma; Deepak Kumar; Shweta Sehrawat; Dinesh Kumar; Sumit Kumar

55

Dissolution improvement and solubility enhancement of two tumor-associated enzyme inhibitors via the formation of eutectic mixtures

Journal of Pharmaceutical Sciences 114(9) (2025)

Chenchen Wang; Xingyin Wang; Chaoyang Yin; Lanting Gao; Jie He; Guisen Zhang; Jian Zhang; Chao Hao; Tao Zhuang

56

Application of cosolvency and cocrystallization approach to enhance acyclovir solubility

BMC Chemistry 19(1) (2025)

Elham Azad Khiabani; Abolghasem Jouyban; Anahita Fathi Azarbayjani

57

Development of β‐Cyclodextrin‐Based Nanofiber Inclusion Complexes for Enhanced Solubility and Controlled Release of Nitazoxanide

ChemistrySelect 10(32) (2025)

Naushad Ahmad; Sonaimuthu Mohandoss; Kuppu Sakthi Velu; Ramachandran Srinivasan; Prasanta Roy; Prathap Somu

58

Interaction of linezolid-bound magnetic iron oxide nanoparticle to β-cyclodextrin/DNA

Journal of Molecular Liquids 438 (2025)

Sameena Yousuf; Israel V.M.V. Enoch

59

Lactose based crystalline solid dispersions to enhance ibuprofen solubility via hot-melt extrusion: A design of experiments approach

Carbohydrate Polymer Technologies and Applications 14 (2026)

Nagarjuna Narala; Siva Ram Munnangi; Srikanth Baisa; Preethi Lakkala; Prateek Uttreja; Indrajeet Karnik; Sagar Narala; Sateesh Kumar Vemula; Michael A. Repka

61

Recent Patents on Solid Dispersions Emphasize Promising Benefits in Solubility Enhancement of Poorly Water-soluble Drugs

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Manisha Saini; Shailendra Bhatt; Harish Dureja; Neeta Solanki

62

Solubility enhancement of Cefpodoxime acid by aqueous solution of paracetamol through acoustical, polarizable continuum model and antimicrobial activity studies

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S.G. Mohammed Hussain; Rathinavelu Kumar; T. Lalitha Sree; Perumal Balu; Venu Kannappan

64

FORMULATION AND CHARACTERIZATION OF ISRADIPINE SOLID DISPERSION WITH ENHANCED SOLUBILITY

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66

A Comparative Study to Examine the Effects of Topical Vinpocetine and Tacrolimus on Induced Atopic Dermatitis in Mice.

Tikrit Journal of Pharmaceutical Sciences 17(2) (2023)

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67

PREPARATION OF SPRAY-DRIED MULTICOMPONENT CRYSTALS OF TRIMETHOPRIM-MANDELIC ACID AND ITS PHYSICOCHEMICAL CHARACTERIZATION

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68

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Deniz Ajabi Zareian; Kobra Rostamizadeh; Nastaran Hashemzadeh; Hossein Danafar; Abolghasem Jouyban

69

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Esther Okafor; Mercy Bella-Omunagbe; Temitope Elugbadebo; Titilope M. Dokunmu; Ezekiel Femi Adebiyi

70

Advanced Techniques in Solubility Enhancement of Poorly Water-Soluble Drugs

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71

ORGANIC ORIGIN GLUCIDES ALDITOLS AS CARRIERS FOR OPTIMIZING SOLUBILIZATION AND DRUG RELEASE

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MOHAMMED A. AMIN; MOSTAFA A. MOHAMED; DALIA A. GABER; HEBA ALI SOLIMAN

72

Enhanced Solubility and Dissolution of Selexipag via β-Cyclodextrin Inclusion Complexes: Formulation and Evaluation

Ars Pharmaceutica (Internet) 67(1) (2025)

Kondi Vanitha; Satya Lakshmi; Prasanna Kumar Desu; Vema Kiran; Battu Srimukhi; Choudary Soujanya

73

Regulatory Considerations of Nanocrystal in Pharmaceutical Sciences

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74

Solubility Enhancement Strategies for Poorly Soluble Drugs: Recent Trends

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75

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Waqar Ahmad; Waqar Ahmad; Hamza Zahid; Maryam; Mir Tanveerul Hassan; Waleed Alam; Khalid Mahmood; Ki‐Duk Song; Mubashir Ahmad

76

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77

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78

Cocristales, una alternativa para potenciar la solubilidad de los fármacos y el desarrollo de nuevos medicamentos

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79

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G. Anusuya; S. Harini; S. Kanshiya; R. Jayasandhiya; Yuvalakshmi Logesan

80

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