OpenCitations
Works that cite this article, indexed by OpenCitations.
Various Aspects of Solid Dispersion Technology: A Review
Research Journal of Pharmacy and Technology (2025)
Deepika Sharma; Deepak Kumar; Shweta Sehrawat; Dinesh Kumar; Sumit Kumar
Cocrystal Engineering-Based Strategies for Enhancing the Permeability of Poorly Permeable APIs
Crystal Growth & Design 25(18) (2025)
Maan Singh; Mayuri P. Sawarkar; Madhukiran R. Dhondale; Dolores R. Serrano; Ashish Kumar Agrawal; Dinesh Kumar
Advanced Techniques in Solubility Enhancement of Poorly Water-Soluble Drugs
Research Journal of Pharmacy and Technology (2025)
Amrita Nayak; Rama Prasad Padhy; Deepak Kumar Bhatta; Gourhari Pal; Bhuneswari Bareha; Aanchal Gupta
Computational Modelling for Formulation Design
Applications of Computational Tools in Drug Design and Development (2025)
Teja Kumar Ponduri; Roja Rani Budha; Deepika Paliwal; Kartheek Siripurapu; Rajasekhar Reddy Alavala; S. N. Koteswara Rao G.
Biofunctional Excipients: Their Emerging Role in Overcoming the Inherent Poor Biopharmaceutical Characteristics of Drugs
Pharmaceutics 17(5) (2025)
Milad Reda Qelliny; Wesam W. Mustafa; Adel Al Fatease; Ali H. Alamri; Raid Alany; Hamdy Abdelkader
Dissolution improvement and solubility enhancement of two tumor-associated enzyme inhibitors via the formation of eutectic mixtures
Journal of Pharmaceutical Sciences 114(9) (2025)
Chenchen Wang; Xingyin Wang; Chaoyang Yin; Lanting Gao; Jie He; Guisen Zhang; Jian Zhang; Chao Hao; Tao Zhuang
Development and Characterization of Polymeric Films Loaded with Terbinafine for Fungal Infection Treatment
Polymers 17(8) (2025)
Gabriela Biliuta; Simona Petronela Gherman; Raluca Ioana Baron; Alexandra Bargan; Lacramioara Ochiuz; Cristina Gabriela Tuchilus; Adrian Florin Spac; Daniela Elena Zavastin
Development and Characterization of an Ibuprofen-Salicylic Acid Co-crystal with Improved Solubility
Journal of Pharmaceutical Innovation 20(2) (2025)
Sonal Dubey; Dheerathi T; Dilip R. Reddy; Manisha Rajou
A Comprehensive Review on Polycaprolactone: A Promising Polymer for Enhancing Drug Bioavailability
Polymer-Plastics Technology and Materials 64(13) (2025)
Swati Dubey; Sanjeev Kumar Patel; Madhulika Pradhan; Krishna Yadav; Sunita Minz
Development of β‐Cyclodextrin‐Based Nanofiber Inclusion Complexes for Enhanced Solubility and Controlled Release of Nitazoxanide
ChemistrySelect 10(32) (2025)
Naushad Ahmad; Sonaimuthu Mohandoss; Kuppu Sakthi Velu; Ramachandran Srinivasan; Prasanta Roy; Prathap Somu
Review: Solid Dispersion Formulation Methods and Applications in Drug Delivery
Current Physical Chemistry 15(2) (2025)
Neelam Sihag; Kavita Bahmani; Samiksha Grewal; Rajni Tanwar; Nisham Rani; Jyoti Malik; Sunita Devi
A single crystal to single crystal solvatomorphic phase transition in cocrystals of pyrimethamine with 4-hydroxybenzoic acid. An experimental and theoretical study
CrystEngComm 27(27) (2025)
Aqsa Bilal; Arshad Mehmood; Sajida Noureen; Maqsood Ahmed
Enhanced solubility of poorly water-soluble drugs in a choline chloride/diethylene glycol deep eutectic solvent: experimental and thermodynamic modeling
Journal of Molecular Liquids 447 (2026)
Reyhaneh Kefayati; Ali Haghtalab
Enhanced Solubility and Dissolution of Selexipag via β-Cyclodextrin Inclusion Complexes: Formulation and Evaluation
Ars Pharmaceutica (Internet) 67(1) (2025)
Kondi Vanitha; Satya B Lakshmi; Kumar Desu Prasanna; Vema Kiran; Battu Srimukhi; Choudary Soujanya
ORGANIC ORIGIN GLUCIDES ALDITOLS AS CARRIERS FOR OPTIMIZING SOLUBILIZATION AND DRUG RELEASE
International Journal of Applied Pharmaceutics (2025)
MOHAMMED A. AMIN; MOSTAFA A. MOHAMED; DALIA A. GABER; HEBA ALI SOLIMAN
Interaction of linezolid-bound magnetic iron oxide nanoparticle to β-cyclodextrin/DNA
Journal of Molecular Liquids 438 (2025)
Sameena Yousuf; Israel V.M.V. Enoch
Cationic surfactants: Fundamental aspects and functionality in the light of petrochemical industry challenges
Journal of Molecular Liquids 439 (2025)
G.A. Gaynanova; L.A. Vasileva; E.A. Romanova; L.Ya. Zakharova; O.G. Sinyashin
Targeting invasion-associated proteins PfSUB2 and PfTRAMP in Plasmodium falciparum: identification of potential inhibitors via molecular docking
BMC Infectious Diseases 25(1) (2025)
Esther. O. Okafor; Mercy Bella-Omunagbe; Temitope Elugbadebo; Titilope M. Dokunmu; Ezekiel Adebiyi
Regulatory Considerations of Nanocrystal in Pharmaceutical Sciences
Nanocrystal Technologies in Biomedical Sciences (2026)
Vasu Peddinti; Shyam Sudhakar Gomte; Devaraj Yallappa; Shruti Patil; Aakanchha Jain
Therapeutic Potential of 2,2′:6′,2″-Terpyridine-Based Au(III), Pt(II), and Mn(II) Complexes against 2D and 3D Human Colorectal Resistant Cancer Cells
Journal of Medicinal Chemistry 68(21) (2025)
Katarzyna Choroba; Barbara Machura; Mateusz Penkala; Karol Erfurt; Sandra Cordeiro; Vanessa Araújo; Edvânia Leopoldo; Rute Lima; Diogo Afonso; Pedro V. Baptista; Alexandra R. Fernandes
A Comprehensive Review of Solubility Enhancement Techniques for Poorly Soluble Drugs
Journal of Solution Chemistry 55(2) (2025)
Rajeswari Saripilli; Dinesh Kumar Sharma
Design Strategies for Improving Oral Bioavailability of Tizanidine: Solid Dispersion Approach
INTERNATIONAL JOURNAL OF DRUG DELIVERY TECHNOLOGY 14(03) (2024)
Manisha . Saini; Suresh . Kumar; Vikas . Jhawat; Rameshwar . Dass
Enhancing the Solubility of Co-Formulated Hydrophobic Drugs by Incorporating Functionalized Nano-Structured Poly Lactic-co-glycolic Acid (nfPLGA) During Co-Precipitation
Pharmaceutics 17(1) (2025)
Mohammad Saiful Islam; Somenath Mitra
CFD modelling and simulations of atomization-based processes for production of drug particles: A review
International Journal of Pharmaceutics 670 (2025)
Mohamad Baassiri; Vivek Ranade; Luis Padrela
A Quaternary Solid Dispersion System for Improving the Solubility of Olaparib
Solids 6(1) (2025)
Tae-Han Yun; Jeong-Gyun Lee; Kyu-Ho Bang; Jung-Hyun Cho; Kyeong-Soo Kim
Oligoethylene Phosphoramidate‐Based Kinase Inhibitor Prodrugs – Solubility, Enzyme Inhibition, and Hydrolysis
Chemistry – A European Journal 31(12) (2025)
Sarah Spiewok; Maximilian Schaefer; Markus Lamla; Yannick Jaritz; Alexander J. C. Kuehne
FORMULATION AND CHARACTERIZATION OF ISRADIPINE SOLID DISPERSION WITH ENHANCED SOLUBILITY
International Journal of Applied Pharmaceutics (2025)
ZAID HADI FAKHRULDEEN; MAZIN THAMIR ABDUL-HASAN
Preparation of Amorphous Probucol with Fluvastatin Sodium Salt and Stability Comparison Studies of Co-amorphous Probucol with Fluvastatin Sodium Salt and Atorvastatin Calcium Trihydrate Salt
Chemical and Pharmaceutical Bulletin 72(12) (2024)
Shinji Oyama; Noriko Ogawa; Toshiya Yasunaga; Hiromitsu Yamamoto
Dissolution methods to discriminate in vitro dissolution of poor water soluble weak base drug using three strategies: Acid modification, solvent evaporation and gastroretentive: Ciprofloxacin HCl case
Journal of Research in Pharmacy 29(1) (2025)
Ahmed Ali Hashim Al Ameri; Masar Basim Mohsin Mohamed
Cocrystals of antibiotics: enhancing antimicrobial efficacy through crystal engineering
Chemical Papers 79(5) (2025)
Amin Alvani; Ali Shayanfar; Raha Kaviani
Principal component analysis (PCA) of bioactive compounds and antioxidant activity of various sample particle sizes of sea urchin shells from coastal area of Lombok Island
Research Journal of Pharmacy and Technology (2024)
Legis Ocktaviana Saputri; Nurhidayati Nurhidayati; Herpan Syafii Harahap; Fitriannisa Faradina Zubaidi; Arina Windri Rivarti; Lina Permatasari
A comprehensive review of green approaches to drug solubility enhancement
Drug Development and Industrial Pharmacy 51(7) (2025)
B. S. Mahesha; F. R. Sheeba; H. K. Deepak
Application of cosolvency and cocrystallization approach to enhance acyclovir solubility
BMC Chemistry 19(1) (2025)
Elham Azad Khiabani; Abolghasem Jouyban; Anahita Fathi Azarbayjani
Development and characterization of furosemide-loaded binary amorphous solid dispersion to enhance solubility and dissolution for pediatric oral administration
Pharmacia 72 (2025)
Mays Fadhil Mohammed-Kadhum; Ghaidaa S. Hameed
Seven New Irbesartan Salts: Significantly Improved Dissolution, Excellent Hygrothermal Stability, and Characteristic Supramolecular Synthons
Crystals 15(4) (2025)
Junxiao Wang; Chuanhua Wu; Menglong Zhang; Lingli Hou; Wei Chen; Dingding Jing; Ying Bao
Choline-Amino Acid-Derived Bio-ionic Liquids for Solubility Enhancement of Zafirlukast
AAPS PharmSciTech 23(5) (2022)
Namrata Gaikwad; Swapna Kudal; Amelia M. Avachat
Recent Patents on Solid Dispersions Emphasize Promising Benefits in Solubility Enhancement of Poorly Water-soluble Drugs
Recent Patents on Nanotechnology 19(2) (2025)
Manisha Saini; Shailender Bhatt; Harish Dureja; Neeta Solanki
A Phosphoramidate Prodrug Platform: One‐Pot Amine Functionalization of Kinase Inhibitors with Oligoethylene Glycol for Improved Water‐Solubility
Chemistry – A European Journal 30(49) (2024)
Sarah Spiewok; Markus Lamla; Maximilian Schaefer; Alexander J. C. Kuehne
Recent developments in the use of nanocrystals to improve bioavailability of APIs
WIREs Nanomedicine and Nanobiotechnology 16(2) (2024)
Yidan Ding; Tongyi Zhao; Jianing Fang; Jiexin Song; Haobo Dong; Jiarui Liu; Sijin Li; Min Zhao
Development and validation of analytical methods for multicomponent crystals of ibuprofen with malic and tartaric acid using spectrophotometry
Journal of Physics: Conference Series 2190(1) (2022)
S P Susilo; S H Pertiwi; A Ainurofiq
Validation of UV spectrophotometric method for ketoprofen multicomponent crystals with malic acid and tartaric acid
Journal of Physics: Conference Series 2190(1) (2022)
C F S Syamdini; I K Muthiah; A Ainurofiq
New salts of teriflunomide (TFM) – Single crystal X-ray and solid state NMR investigation
Solid State Nuclear Magnetic Resonance 122 (2022)
Tomasz Pawlak; Piotr Paluch; Rafał Dolot; Grzegorz Bujacz; Marek J. Potrzebowski
Third-Generation Solid Dispersion Through Lyophilization Enhanced Oral Bioavailability of Resveratrol
ACS Pharmacology & Translational Science 7(3) (2024)
Hugo Almeida; Bárbara Ferreira; Carlos Fernandes-Lopes; Francisca Araújo; Maria João Bonifácio; Teófilo Vasconcelos; Bruno Sarmento
Towards the prediction of drug solubility in binary solvent mixtures at various temperatures using machine learning
Journal of Cheminformatics 16(1) (2024)
Zeqing Bao; Gary Tom; Austin Cheng; Jeffrey Watchorn; Alán Aspuru-Guzik; Christine Allen
Solubility enhancement of caffeine and furosemide using deep eutectic solvents formed by choline chloride and xylitol, citric acid, sorbitol or glucose
Journal of Drug Delivery Science and Technology 79 (2023)
Laura Lomba; Alejandra Polo; Julia Alejandre; Nuria Martínez; Beatriz Giner
Rational and experimental investigation of antihypotensive midodrine-Fe(III) complex: Synthesis, spectroscopy, DFT, biological activity and molecular docking
Journal of Molecular Structure 1311 (2024)
Doaa S. El Sayed; Tarek E. Khalil; Hemmat A. Elbadawy
Sugars and Polyols of Natural Origin as Carriers for Solubility and Dissolution Enhancement
Pharmaceutics 15(11) (2023)
Madan Sai Poka; Marnus Milne; Anita Wessels; Marique Aucamp
Solubility behavior of Rosiglitazone in ten pure solvents: Model correlation, thermodynamic calculations, and molecular simulation
Journal of Molecular Liquids 417 (2025)
Xiaojie Zhou; Aoran Xiong; Yuxi Zhen; Yizhen Yan; Xiangyang Zhang
A Scalable Freeze-Dissolving Approach to Prepare Ultrafine Crystals for Inhalation: Mechanism and Validation
Crystal Growth & Design 24(7) (2024)
Shengzheng Guo; Yuechao Cao; Yuxin Zhang; Yan Wang; Zhenguo Gao; Junbo Gong
Solubility enhancement of Cefpodoxime acid by aqueous solution of paracetamol through acoustical, polarizable continuum model and antimicrobial activity studies
Journal of Molecular Liquids 395 (2024)
S.G. Mohammed Hussain; R. Kumar; T. Lalitha Sree; P. Balu; V. Kannappan
Unveiling the role of solubilization of metformin hydrochloride assimilated in nonionic surfactants mediated mixed micellar assemblies
Colloids and Surfaces A: Physicochemical and Engineering Aspects 703 (2024)
Nida Fatima; Muhammad Usman; Amnah Yusaf; Tanveer Hussain Bokhari; Nadia Akram; Saima Rehman; Sajjad Haider; Muhammad Siddiq; Muhammad Ahsan Bhatti; Muhammad Arif Cheema
Examine stability polyvinyl alcohol-stabilized nanosuspensions to overcome the challenge of poor drug solubility utilizing molecular dynamic simulation
Scientific Reports 14(1) (2024)
Sedigheh Abdollahi; Heidar Raissi; Farzaneh Farzad
Emerging role of nanocrystals in pharmaceutical applications: A review of regulatory aspects and drug development process
Applied Materials Today 40 (2024)
Padakanti Sandeep Chary; Samia Shaikh; Valamla Bhavana; Naveen Rajana; Ravindra Vasave; Neelesh Kumar Mehra
Design of Etched- and Functionalized-Halloysite/Meloxicam Hybrids: A Tool for Enhancing Drug Solubility and Dissolution Rate
Pharmaceutics 16(3) (2024)
Valeria Friuli; Claudia Urru; Chiara Ferrara; Debora Maria Conti; Giovanna Bruni; Lauretta Maggi; Doretta Capsoni
Microwave-assisted, sulfhydryl-modified β-cyclodextrin-silymarin inclusion complex: A diverse approach to improve oral drug bioavailability via enhanced mucoadhesion and permeation
Carbohydrate Polymers 348 (2025)
Shumaila Arshad; Syed Atif Raza; Alamgeer; Syed Nasir Abbas Bukhari; Nasser F. Alotaibi; Naveed Ahmad; Hafiz Muhammad Irfan; Arshad Mahmood; Mulazim Hussain Asim
Recent advancements toward the incremsent of drug solubility using environmentally-friendly supercritical CO2: a machine learning perspective
Frontiers in Medicine 11 (2024)
Jawaher Abdullah Alamoudi
Novel Biphasic In Vitro Dissolution Method Correctly Predicts the Oral Bioavailability of Curcumin in Humans
Journal of Agricultural and Food Chemistry 71(42) (2023)
Marvin Benedikt Brenner; Sandra Flory; Matthias Wüst; Jan Frank; Karl Wagner
Low-melting mixture solvents as novel solubilizing agents: Improving tolvaptan formulation and therapeutic efficacy
Journal of Molecular Liquids 414 (2024)
Xiuxiu Huang; Wenqing Dong; Xiao Luo; Lu Xu; Dongzhi Yang; Yinan Wang
PREPARATION OF SPRAY-DRIED MULTICOMPONENT CRYSTALS OF TRIMETHOPRIM-MANDELIC ACID AND ITS PHYSICOCHEMICAL CHARACTERIZATION
International Journal of Applied Pharmaceutics (2024)
LILI FITRIANI; DENANDA SHINTANIA; HENDRIZAL USMAN; USWATUL HASANAH; ERIZAL ZAINI
The Effect of the Particle Size Reduction on the Biorelevant Solubility and Dissolution of Poorly Soluble Drugs with Different Acid-Base Character
Pharmaceutics 15(1) (2023)
Dóra Csicsák; Rita Szolláth; Szabina Kádár; Rita Ambrus; Csilla Bartos; Emese Balogh; István Antal; István Köteles; Petra Tőzsér; Vivien Bárdos; Péter Horváth; Enikő Borbás; Krisztina Takács-Novák; Bálint Sinkó; Gergely Völgyi
Mathematical optimization and prediction of Febuxostat xanthine oxidase inhibitor solubility through supercritical CO2 system using machine-learning approach
Journal of Molecular Liquids 387 (2023)
Umme Hani; Zainab Ali Bu Sinnah; Ahmad J. Obaidullah; Jowaher Alanazi; Muteb Alanazi; Tareq Nafea Alharby; Ahmed Abdullah Al Awadh; Ahmed A. Lahiq
Ibuprofen solubility and cytotoxic study of deep eutectic solvents formed by xylitol, choline chloride and water
Journal of Drug Delivery Science and Technology 82 (2023)
Laura Lomba; Mª Pilar Garralaga; Álvaro Werner; Beatriz Giner; Pedro M. Baptista; Natalia Sánchez-Romero
Enhancing the dissolution and bacteriostatic activity of trimethoprim through salt formation
CrystEngComm 25(23) (2023)
Xingchen Hu; Yuntian Xiao; Luguang Qi; Yunhe Bai; Ying Sun; Yang Ye; Chuang Xie
Physical stability and dissolution of ketoprofen nanosuspension formulation: Polyvinylpyrrolidone and Tween 80 as stabilizers
Pharmacia 70(1) (2023)
Tengku Ismanelly Hanum; Azizah Nasution; Sumaiyah Sumaiyah; Hakim Bangun
A Comparison of Spray-Drying and Co-Precipitation for the Generation of Amorphous Solid Dispersions (ASDs) of Hydrochlorothiazide and Simvastatin
Journal of Pharmaceutical Sciences 112(8) (2023)
Monika Myślińska; Michael W. Stocker; Steven Ferguson; Anne Marie Healy
Deep eutectic solvents based on sugars for oral applications
European Journal of Pharmaceutics and Biopharmaceutics 191 (2023)
Laura Lomba; Alejandra Polo; Álvaro Werner; Carlos Lafuente; Beatriz Giner
Study of sertraline solubility, solvent effect, and modeling in the aqueous mixtures of dimethyl sulfoxide or diethylene glycol monoethyl ether at several temperatures and its use in the formulation of nanosuspensions
Journal of Drug Delivery Science and Technology 99 (2024)
Deniz Ajabi Zareian; Kobra Rostamizadeh; Nastaran Hashemzadeh; Hossein Danafar; Abolghasem Jouyban
Experimental screening and molecular dynamics simulation study on wetting agent in dry suspension
Journal of Drug Delivery Science and Technology 95 (2024)
Minfang Feng; Yuting Tian; Yingying Zhang; Cuiting Yang; Xinhui Peng; Shuai Cen; Mengke Sheng; Zhixun Li; Qing Zhou; Xingxing Dai; Xinyuan Shi
Nanocrystals: A Deep Insight into Formulation Aspects, Stabilization Strategies, and Biomedical Applications
Recent Patents on Nanotechnology 17(4) (2023)
Parijat Pandey; Deepika Purohit; Shivkant Sharma; Avneet Kaur Lamba; Sapna Saini; Neha Minocha; Neelam Vashist; Dhirender Kaushik