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73 resultsUpdated October 20, 2026
1

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Deepika Sharma; Deepak Kumar; Shweta Sehrawat; Dinesh Kumar; Sumit Kumar

2

Cocrystal Engineering-Based Strategies for Enhancing the Permeability of Poorly Permeable APIs

Crystal Growth & Design 25(18) (2025)

Maan Singh; Mayuri P. Sawarkar; Madhukiran R. Dhondale; Dolores R. Serrano; Ashish Kumar Agrawal; Dinesh Kumar

3

Advanced Techniques in Solubility Enhancement of Poorly Water-Soluble Drugs

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Amrita Nayak; Rama Prasad Padhy; Deepak Kumar Bhatta; Gourhari Pal; Bhuneswari Bareha; Aanchal Gupta

4

Computational Modelling for Formulation Design

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Teja Kumar Ponduri; Roja Rani Budha; Deepika Paliwal; Kartheek Siripurapu; Rajasekhar Reddy Alavala; S. N. Koteswara Rao G.

5

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Milad Reda Qelliny; Wesam W. Mustafa; Adel Al Fatease; Ali H. Alamri; Raid Alany; Hamdy Abdelkader

6

Dissolution improvement and solubility enhancement of two tumor-associated enzyme inhibitors via the formation of eutectic mixtures

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Chenchen Wang; Xingyin Wang; Chaoyang Yin; Lanting Gao; Jie He; Guisen Zhang; Jian Zhang; Chao Hao; Tao Zhuang

7

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Gabriela Biliuta; Simona Petronela Gherman; Raluca Ioana Baron; Alexandra Bargan; Lacramioara Ochiuz; Cristina Gabriela Tuchilus; Adrian Florin Spac; Daniela Elena Zavastin

8

Development and Characterization of an Ibuprofen-Salicylic Acid Co-crystal with Improved Solubility

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Sonal Dubey; Dheerathi T; Dilip R. Reddy; Manisha Rajou

9

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Swati Dubey; Sanjeev Kumar Patel; Madhulika Pradhan; Krishna Yadav; Sunita Minz

10

Development of β‐Cyclodextrin‐Based Nanofiber Inclusion Complexes for Enhanced Solubility and Controlled Release of Nitazoxanide

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Naushad Ahmad; Sonaimuthu Mohandoss; Kuppu Sakthi Velu; Ramachandran Srinivasan; Prasanta Roy; Prathap Somu

11

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Neelam Sihag; Kavita Bahmani; Samiksha Grewal; Rajni Tanwar; Nisham Rani; Jyoti Malik; Sunita Devi

14

Enhanced Solubility and Dissolution of Selexipag via β-Cyclodextrin Inclusion Complexes: Formulation and Evaluation

Ars Pharmaceutica (Internet) 67(1) (2025)

Kondi Vanitha; Satya B Lakshmi; Kumar Desu Prasanna; Vema Kiran; Battu Srimukhi; Choudary Soujanya

15

ORGANIC ORIGIN GLUCIDES ALDITOLS AS CARRIERS FOR OPTIMIZING SOLUBILIZATION AND DRUG RELEASE

International Journal of Applied Pharmaceutics (2025)

MOHAMMED A. AMIN; MOSTAFA A. MOHAMED; DALIA A. GABER; HEBA ALI SOLIMAN

16

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Sameena Yousuf; Israel V.M.V. Enoch

17

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Journal of Molecular Liquids 439 (2025)

G.A. Gaynanova; L.A. Vasileva; E.A. Romanova; L.Ya. Zakharova; O.G. Sinyashin

18

Targeting invasion-associated proteins PfSUB2 and PfTRAMP in Plasmodium falciparum: identification of potential inhibitors via molecular docking

BMC Infectious Diseases 25(1) (2025)

Esther. O. Okafor; Mercy Bella-Omunagbe; Temitope Elugbadebo; Titilope M. Dokunmu; Ezekiel Adebiyi

19

Regulatory Considerations of Nanocrystal in Pharmaceutical Sciences

Nanocrystal Technologies in Biomedical Sciences (2026)

Vasu Peddinti; Shyam Sudhakar Gomte; Devaraj Yallappa; Shruti Patil; Aakanchha Jain

20

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21

A Comprehensive Review of Solubility Enhancement Techniques for Poorly Soluble Drugs

Journal of Solution Chemistry 55(2) (2025)

Rajeswari Saripilli; Dinesh Kumar Sharma

22

Design Strategies for Improving Oral Bioavailability of Tizanidine: Solid Dispersion Approach

INTERNATIONAL JOURNAL OF DRUG DELIVERY TECHNOLOGY 14(03) (2024)

Manisha . Saini; Suresh . Kumar; Vikas . Jhawat; Rameshwar . Dass

24

CFD modelling and simulations of atomization-based processes for production of drug particles: A review

International Journal of Pharmaceutics 670 (2025)

Mohamad Baassiri; Vivek Ranade; Luis Padrela

25

A Quaternary Solid Dispersion System for Improving the Solubility of Olaparib

Solids 6(1) (2025)

Tae-Han Yun; Jeong-Gyun Lee; Kyu-Ho Bang; Jung-Hyun Cho; Kyeong-Soo Kim

26

Oligoethylene Phosphoramidate‐Based Kinase Inhibitor Prodrugs – Solubility, Enzyme Inhibition, and Hydrolysis

Chemistry – A European Journal 31(12) (2025)

Sarah Spiewok; Maximilian Schaefer; Markus Lamla; Yannick Jaritz; Alexander J. C. Kuehne

27

FORMULATION AND CHARACTERIZATION OF ISRADIPINE SOLID DISPERSION WITH ENHANCED SOLUBILITY

International Journal of Applied Pharmaceutics (2025)

ZAID HADI FAKHRULDEEN; MAZIN THAMIR ABDUL-HASAN

30

Cocrystals of antibiotics: enhancing antimicrobial efficacy through crystal engineering

Chemical Papers 79(5) (2025)

Amin Alvani; Ali Shayanfar; Raha Kaviani

31

Principal component analysis (PCA) of bioactive compounds and antioxidant activity of various sample particle sizes of sea urchin shells from coastal area of Lombok Island

Research Journal of Pharmacy and Technology (2024)

Legis Ocktaviana Saputri; Nurhidayati Nurhidayati; Herpan Syafii Harahap; Fitriannisa Faradina Zubaidi; Arina Windri Rivarti; Lina Permatasari

32

A comprehensive review of green approaches to drug solubility enhancement

Drug Development and Industrial Pharmacy 51(7) (2025)

B. S. Mahesha; F. R. Sheeba; H. K. Deepak

33

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35

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36

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AAPS PharmSciTech 23(5) (2022)

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37

Recent Patents on Solid Dispersions Emphasize Promising Benefits in Solubility Enhancement of Poorly Water-soluble Drugs

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Manisha Saini; Shailender Bhatt; Harish Dureja; Neeta Solanki

38

A Phosphoramidate Prodrug Platform: One‐Pot Amine Functionalization of Kinase Inhibitors with Oligoethylene Glycol for Improved Water‐Solubility

Chemistry – A European Journal 30(49) (2024)

Sarah Spiewok; Markus Lamla; Maximilian Schaefer; Alexander J. C. Kuehne

39

Recent developments in the use of nanocrystals to improve bioavailability of APIs

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Yidan Ding; Tongyi Zhao; Jianing Fang; Jiexin Song; Haobo Dong; Jiarui Liu; Sijin Li; Min Zhao

41

Validation of UV spectrophotometric method for ketoprofen multicomponent crystals with malic acid and tartaric acid

Journal of Physics: Conference Series 2190(1) (2022)

C F S Syamdini; I K Muthiah; A Ainurofiq

42

New salts of teriflunomide (TFM) – Single crystal X-ray and solid state NMR investigation

Solid State Nuclear Magnetic Resonance 122 (2022)

Tomasz Pawlak; Piotr Paluch; Rafał Dolot; Grzegorz Bujacz; Marek J. Potrzebowski

43

Third-Generation Solid Dispersion Through Lyophilization Enhanced Oral Bioavailability of Resveratrol

ACS Pharmacology & Translational Science 7(3) (2024)

Hugo Almeida; Bárbara Ferreira; Carlos Fernandes-Lopes; Francisca Araújo; Maria João Bonifácio; Teófilo Vasconcelos; Bruno Sarmento

44

Towards the prediction of drug solubility in binary solvent mixtures at various temperatures using machine learning

Journal of Cheminformatics 16(1) (2024)

Zeqing Bao; Gary Tom; Austin Cheng; Jeffrey Watchorn; Alán Aspuru-Guzik; Christine Allen

45

Solubility enhancement of caffeine and furosemide using deep eutectic solvents formed by choline chloride and xylitol, citric acid, sorbitol or glucose

Journal of Drug Delivery Science and Technology 79 (2023)

Laura Lomba; Alejandra Polo; Julia Alejandre; Nuria Martínez; Beatriz Giner

47

Sugars and Polyols of Natural Origin as Carriers for Solubility and Dissolution Enhancement

Pharmaceutics 15(11) (2023)

Madan Sai Poka; Marnus Milne; Anita Wessels; Marique Aucamp

48

Solubility behavior of Rosiglitazone in ten pure solvents: Model correlation, thermodynamic calculations, and molecular simulation

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Xiaojie Zhou; Aoran Xiong; Yuxi Zhen; Yizhen Yan; Xiangyang Zhang

49

A Scalable Freeze-Dissolving Approach to Prepare Ultrafine Crystals for Inhalation: Mechanism and Validation

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50

Solubility enhancement of Cefpodoxime acid by aqueous solution of paracetamol through acoustical, polarizable continuum model and antimicrobial activity studies

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S.G. Mohammed Hussain; R. Kumar; T. Lalitha Sree; P. Balu; V. Kannappan

51

Unveiling the role of solubilization of metformin hydrochloride assimilated in nonionic surfactants mediated mixed micellar assemblies

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53

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54

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55

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57

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58

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59

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60

The Effect of the Particle Size Reduction on the Biorelevant Solubility and Dissolution of Poorly Soluble Drugs with Different Acid-Base Character

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61

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62

Ibuprofen solubility and cytotoxic study of deep eutectic solvents formed by xylitol, choline chloride and water

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63

Enhancing the dissolution and bacteriostatic activity of trimethoprim through salt formation

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65

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66

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