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10 resultsUpdated October 24, 2026
1

Lead Optimization of a Butyrylcholinesterase Inhibitor for the Treatment of Alzheimer’s Disease

Journal of Medicinal Chemistry 68(11) (2025)

Urban Košak; Nika Strašek Benedik; Damijan Knez; Simon Žakelj; Jurij Trontelj; Anja Hafner Pišlar; Selena Horvat; Aljoša Bolje; Neža Žnidaršič; Neža Grgurevič; Tanja Švara; Jakob Kljun; Anna Skrzypczak-Wiercioch; Bingbing Lv; Yucheng Xiong; Qinjie Wang; Rui Bian; Jikuan Shao; José Dias; Florian Nachon; Xavier Brazzolotto; Jure Stojan; Haopeng Sun; Kinga Sałat; Stanislav Gobec

2

N-Propargylpyrrolidine-based butyrylcholinesterase and monoamine oxidase inhibitors

Chemico-Biological Interactions 420 (2025)

Urban Košak; Damijan Knez; Anja Hafner Pišlar; Selena Horvat; Simon Žakelj; Alexandre Igert; José Dias; Florian Nachon; Xavier Brazzolotto; Stanislav Gobec

3

Dose-Dependent Dissociation of Pro-cognitive Effects of Donepezil on Attention and Cognitive Flexibility in Rhesus Monkeys

Biological Psychiatry Global Open Science 3(1) (2021)

Seyed A. Hassani; Sofia Lendor; Adam R. Neumann; Kanchan Sinha Roy; Kianoush Banaie Boroujeni; Kari L. Hoffman; Janusz B. Pawliszyn; Thilo Womelsdorf

4

Analgesic and preventive effects of donepezil in animal models of chemotherapy-induced peripheral neuropathy: Involvement of spinal muscarinic acetylcholine M2 receptors

Biomedicine & Pharmacotherapy 149 (2022)

Marie Selvy; Catherine Mattevi; Cristelle Dalbos; Youssef Aissouni; Eric Chapuy; Pierre-Yves Martin; Aurore Collin; Damien Richard; Charles Dumontet; Jérôme Busserolles; Sakahlé Condé; David Balayssac

5

Antioxidant and Anticholinesterase Properties of the Aqueous Extract of Balanites aegyptiaca L. Delile Fruit Pulp on Monosodium Glutamate-Induced Excitotoxicity in Swiss Mice

Evidence-based Complementary and Alternative Medicine 2022 (2022)

Parfait Bouvourné; Galba Jean Beppe; Roger Ponka; Ngatanko Abaïssou Hervé Hervé; Balbine Kamleu Nkwingwa; Guillaume Woumitna Camdi; Guedang Nyayi Simon Désiré; Jorelle Linda Damo Kamda; Kenko Djoumessie Léa Blondelle; Germain Sotoing Taïwé

6

Drug Distribution in Brain and Cerebrospinal Fluids in Relation to IC50 Values in Aging and Alzheimer’s Disease, Using the Physiologically Based LeiCNS-PK3.0 Model

Pharmaceutical Research 39(7) (2022)

Mohammed A. A. Saleh; Julia S. Bloemberg; Jeroen Elassaiss‐Schaap; Elizabeth C. M. de Lange

7

The measured CSF/plasma donepezil concentration ratio but not individually measured CSF and plasma concentrations significantly increase over 24 h after donepezil treatment in patients with Alzheimer’s disease

Biomedicine & Pharmacotherapy 159 (2023)

Martin Vališ; Alžběta Dlabková; Jakub Hort; Francesco Angelucci; Jaroslav Pejchal; Kamil Kuča; Zbyšek Pavelek; Jana Žďárová Karasová; Michal Novotný

10

Rapid HPLC-Based ADME Profiling of Novel Donepezil and Rivastigmine Analogues for Potential Application in Alzheimer’s Disease

ACS Omega 11(41) (2026)

Stefan Simić; Rosalba Leuci; Marianne Pirker; Predrag Kalaba; Judith Wackerlig; Luca Piemontese; Thierry Langer