Design and Synthesis of New Imidazole Derivatives of Captopril

Authors

Mohammad Hassan Houshdar Tehrani1,*, Afshin Zarghi1, Laleh Erfani Jabarian1
1Department of Medicinal Chemistry, School of Pharmacy, Shaheed Beheshti University of Medical Sciences and Health Services, Tehran, Iran
*Corresponding Author: Department of Medicinal Chemistry, School of Pharmacy, Shaheed Beheshti University of Medical Sciences and Health Services, Tehran, Iran. Email:[email protected]

Iranian Journal of Pharmaceutical Research:Vol. 4, issue 1; 37-41
Published online:Nov 20, 2010
Article type:Research Article
Received:May 01, 2004
Accepted:Mar 01, 2005
How to Cite:Houshdar Tehrani MH, Zarghi A, Erfani Jabarian L. Design and Synthesis of New Imidazole Derivatives of Captopril. Iran J Pharm Res. 2022;4(1):e128225. doi: https://doi.org/10.22037/ijpr.2010.615

Abstract

A new series of alkylthio imidazole analogues of captopril, an ACE inhibitor used in the treatment of hypertension, was designed and synthesized in order to obtain agents more active than captopril with less side effects. All the compounds thus prepared were purified and characterized by IR, NMR and Mass analytical instruments.

Copyright

© 2022, Author(s). This open-access article is available under the Creative Commons Attribution 4.0 (CC BY 4.0) International License (https://creativecommons.org/licenses/by/4.0/), which allows for unrestricted use, distribution, and reproduction in any medium, provided that the original work is properly cited.

Similar Articles

31
Dec
2018

Novel Group of Imidazole Derivatives as Atypical Selective Cyclooxygenase-2 Inhibitors: Design, Synthesis and Biological Evaluation

Azin Kiani,
Elham Rezaee,
Sayyed Abbas Tabatabai

Kiani A, Rezaee E, Tabatabai SA. Novel Group of Imidazole Derivatives as Atypical Selective Cyclooxygenase-2 Inhibitors: Design, Synthesis and Biological Evaluation. Iran J Pharm Res. 2018;17(Suppl2):e126099. doi: https://doi.org/10.22037/ijpr.2018.2367

30
Apr
2014

N-(5-Mercapto-1,3,4-Thiadiazol-2-yl)-2-Phenylacetamide Derivatives: Synthesis and In-vitro Cytotoxicity Evaluation as Potential Anticancer Agents

Ahmad Mohammadi-Farani,
Neda Heidarian,
Alireza Aliabadi

Mohammadi-Farani A, Heidarian N, Aliabadi A. N-(5-Mercapto-1,3,4-Thiadiazol-2-yl)-2-Phenylacetamide Derivatives: Synthesis and In-vitro Cytotoxicity Evaluation as Potential Anticancer Agents. Iran J Pharm Res. 2014;13(2):e125547. doi: https://doi.org/10.22037/ijpr.2014.1503

31
Mar
2016

Synthesis of Some Spiro Indeno[1,2-b]pyrido[2,3-d]Pyrimidine-5,3′-Indolines as New Urease Inhibitors

Ghodsi Mohammadi Ziarani,
Shima Asadi,
Alireza Badiei,
Amirhossein Sharifi,
Massoud Amanlou

Mohammadi Ziarani G, Asadi S, Badiei A, Sharifi A, Amanlou M. Synthesis of Some Spiro Indeno[1,2-b]pyrido[2,3-d]Pyrimidine-5,3′-Indolines as New Urease Inhibitors. Iran J Pharm Res. 2016;15(Suppl):e125079. doi: https://doi.org/10.22037/ijpr.2016.1806

31
Oct
2015

Design, Synthesis and Evaluation of Antitubercular Activity of Novel Dihydropyridine Containing Imidazolyl Substituent

Maryam Iman,
Asghar Davood,
Golnoush Dehqani,
Mahboubeh Lotfinia,
Soroush Sardari,
Parisa Azerang
,et al.

Iman M, Davood A, Dehqani G, Lotfinia M, Sardari S, et al. Design, Synthesis and Evaluation of Antitubercular Activity of Novel Dihydropyridine Containing Imidazolyl Substituent. Iran J Pharm Res. 2015;14(4):e125381. doi: https://doi.org/10.22037/ijpr.2015.1744

20
Nov
2010

Synthesis and Antimicrobial Activity of Some New Isatin Derivatives

Ankur Patel,
Sanjaykumar Bari,
Gokul Talele,
Jitendra Patel,
Manda Sarangapani

Patel A, Bari S, Talele G, Patel J, Sarangapani M. Synthesis and Antimicrobial Activity of Some New Isatin Derivatives. Iran J Pharm Res. 2022;5(4):e128295. doi: https://doi.org/10.22037/ijpr.2010.685

More by these authors

Mohammad Hassan Houshdar TehraniPubMedScholar
Afshin ZarghiPubMedScholar
Laleh Erfani JabarianPubMedScholar
Share
Cited by
Metrics